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Studies of proline conformational dynamics in IDPs by C-detected cross-correlated NMR relaxation.

2023 Journal of magnetic resonance (San Diego, Calif. : 1997);354:107539.
PMID:  37632987

Schiavina Marco, Konrat Ruth, Ceccolini Irene, Mateos Borja, Konrat Robert, Felli Isabella C, Pierattelli Roberta

Non-uniform sampling of similar NMR spectra and its application to studies of the interaction between alpha-synuclein and liposomes.

2023 Journal of biomolecular NMR;77(4):149, 163, 149-163.
PMID:  37237169

Shchukina Alexandra, Schwarz Thomas C, Nowakowski Michał, Konrat Robert, Kazimierczuk Krzysztof

Crucial neuroprotective roles of the metabolite BH4 in dopaminergic neurons.

2023 bioRxiv : the preprint server for biology
PMID:  37214873

Cronin Shane J F, Yu Weonjin, Hale Ashley, Licht-Mayer Simon, Crabtree Mark J, Korecka Joanna A, Tretiakov Evgenii O, Sealey-Cardona Marco, Somlyay Mate, Onji Masahiro, An Meilin, Fox Jesse D, Turnes Bruna Lenfers, Gomez-Diaz Carlos, da Luz Scheffer Débora, Cikes Domagoj, Nagy Vanja, Weidinger Adelheid, Wolf Alexandra, Reither Harald, Chabloz Antoine, Kavirayani Anoop, Rao Shuan, Andrews Nick, Latremoliere Alban, Costigan Michael, Douglas Gillian, Freitas Fernando Cini, Pifl Christian, Walz Roger, Konrat Robert, Mahad Don J, Koslov Andrey V, Latini Alexandra, Isacson Ole, Harkany Tibor, Hallett Penelope J, Bagby Stefan, Woolf Clifford J, Channon Keith M, Je Hyunsoo Shawn, Penninger Josef M

Early intervention with azelastine nasal spray may reduce viral load in SARS-CoV-2 infected patients.

2023 Scientific reports;13(1):6839.
PMID:  37100830

Klussmann Jens Peter, Grosheva Maria, Meiser Peter, Lehmann Clara, Nagy Eszter, Szijártó Valéria, Nagy Gábor, Konrat Robert, Flegel Michael, Holzer Frank, Groß Dorothea, Steinmetz Charlotte, Scherer Barbara, Gruell Henning, Schlotz Maike, Klein Florian, de Aragão Paula Aguiar, Morr Henning, Al Saleh Helal, Bilstein Andreas, Russo Belisa, Müller-Scholtz Susanne, Acikel Cengizhan, Sahin Hacer, Werkhäuser Nina, Allekotte Silke, Mösges Ralph

High-resolution structural information of membrane-bound α-synuclein provides insight into the MoA of the anti-Parkinson drug UCB0599.

2023 Proceedings of the National Academy of Sciences of the United States of America;120(15):e2201910120.
PMID:  37027427

Schwarz Thomas C, Beier Andreas, Ledolter Karin, Gossenreiter Thomas, Höfurthner Theresa, Hartl Markus, Baker Terry S, Taylor Richard J, Konrat Robert

The Anti-Histamine Azelastine, Identified by Computational Drug Repurposing, Inhibits Infection by Major Variants of SARS-CoV-2 in Cell Cultures and Reconstituted Human Nasal Tissue.

2022 Frontiers in pharmacology;13:861295.
PMID:  35846988

Konrat Robert, Papp Henrietta, Kimpel Janine, Rössler Annika, Szijártó Valéria, Nagy Gábor, Madai Mónika, Zeghbib Safia, Kuczmog Anett, Lanszki Zsófia, Gesell Tanja, Helyes Zsuzsanna, Kemenesi Gábor, Jakab Ferenc, Nagy Eszter

Long-range structural preformation in yes-associated protein precedes encounter complex formation with TEAD.

2022 iScience;25(4):104099.
PMID:  35378854

Feichtinger Michael, Beier Andreas, Migotti Mario, Schmid Matthias, Bokhovchuk Fedir, Chène Patrick, Konrat Robert

Detecting anisotropic segmental dynamics in disordered proteins by cross-correlated spin relaxation.

2021 Magnetic resonance (Gottingen, Germany);2(2):557, 569, 557-569.
PMID:  37905226

Kauffmann Clemens, Ceccolini Irene, Kontaxis Georg, Konrat Robert

A Step toward NRF2-DNA Interaction Inhibitors by Fragment-Based NMR Methods.

2021 ChemMedChem;16(23):3576, 3587, 3576-3587.
PMID:  34524728

Brüschweiler Sven, Fuchs Julian E, Bader Gerd, McConnell Darryl B, Konrat Robert, Mayer Moriz

Association between Predicted Effects of Missense Variants on Protein Conformation and Their Phenotypic Presentation as Li-Fraumeni Syndrome or Hereditary Breast Cancer.

2021 International journal of molecular sciences;22(12)
PMID:  34198491

Liu Yaxuan, Axell Olga, van Leeuwen Tom, Konrat Robert, Kharaziha Pedram, Larsson Catharina, Wright Anthony P H, Bajalica-Lagercrantz Svetlana

On-Cell NMR Contributions to Membrane Receptor Binding Characterization.

2021 ChemPlusChem;86(6):938, 945, 938-945.
PMID:  34160899

Höfurthner Theresa, Mateos Borja, Konrat Robert

Order from disorder in the sarcomere: FATZ forms a fuzzy but tight complex and phase-separated condensates with α-actinin.

2021 Science advances(22)
PMID:  34049882

Sponga Antonio, Arolas Joan L, Schwarz Thomas C, Jeffries Cy M, Rodriguez Chamorro Ariadna, Kostan Julius, Ghisleni Andrea, Drepper Friedel, Polyansky Anton, De Almeida Ribeiro Euripedes, Pedron Miriam, Zawadzka-Kazimierczuk Anna, Mlynek Georg, Peterbauer Thomas, Doto Pierantonio, Schreiner Claudia, Hollerl Eneda, Mateos Borja, Geist Leonhard, Faulkner Georgine, Kozminski Wiktor, Svergun Dmitri I, Warscheid Bettina, Zagrovic Bojan, Gautel Mathias, Konrat Robert, Djinović-Carugo Kristina

Binding Mode Characterization of Osteopontin on Hydroxyapatite by Solution NMR Spectroscopy.

2021 Chembiochem : a European journal of chemical biology;22(13):2300, 2305, 2300-2305.
PMID:  33914399

Holzinger Julian, Kotisch Harald, Richter Klaus W, Konrat Robert

Hyperphosphorylation of Human Osteopontin and Its Impact on Structural Dynamics and Molecular Recognition.

2021 Biochemistry;60(17):1347, 1355, 1347-1355.
PMID:  33876640

Mateos Borja, Holzinger Julian, Conrad-Billroth Clara, Platzer Gerald, Żerko Szymon, Sealey-Cardona Marco, Anrather Dorothea, Koźmiński Wiktor, Konrat Robert

Molecular basis of F-actin regulation and sarcomere assembly via myotilin.

2021 PLoS biology(4)
PMID:  33844684

Kostan Julius, Pavšič Miha, Puž Vid, Schwarz Thomas C, Drepper Friedel, Molt Sibylle, Graewert Melissa Ann, Schreiner Claudia, Sajko Sara, van der Ven Peter F M, Onipe Adekunle, Svergun Dmitri I, Warscheid Bettina, Konrat Robert, Fürst Dieter O, Lenarčič Brigita, Djinović-Carugo Kristina

Cosolute modulation of protein oligomerization reactions in the homeostatic timescale.

2021 Biophysical journal;120(10):2067, 2077, 2067-2077.
PMID:  33794151

Mateos Borja, Bernardo-Seisdedos Ganeko, Dietrich Valentin, Zalba Nicanor, Ortega Gabriel, Peccati Francesca, Jiménez-Osés Gonzalo, Konrat Robert, Tollinger Martin, Millet Oscar

Membrane Interactions of α-Synuclein Revealed by Multiscale Molecular Dynamics Simulations, Markov State Models, and NMR.

2021 The journal of physical chemistry. B;125(11):2929, 2941, 2929-2941.
PMID:  33719460

Amos Sarah-Beth T A, Schwarz Thomas C, Shi Jiye, Cossins Benjamin P, Baker Terry S, Taylor Richard J, Konrat Robert, Sansom Mark S P

Using Cross-Correlated Spin Relaxation to Characterize Backbone Dihedral Angle Distributions of Flexible Protein Segments.

2021 Chemphyschem : a European journal of chemical physics and physical chemistry;22(1):18, 28, 18-28.
PMID:  33119214

Kauffmann Clemens, Zawadzka-Kazimierczuk Anna, Kontaxis Georg, Konrat Robert

Temperature as an Extra Dimension in Multidimensional Protein NMR Spectroscopy.

2021 Chemistry (Weinheim an der Bergstrasse, Germany);27(5):1753, 1767, 1753-1767.
PMID:  32985764

Shchukina Alexandra, Małecki Paweł, Mateos Borja, Nowakowski Michał, Urbańczyk Mateusz, Kontaxis Georg, Kasprzak Paweł, Conrad-Billroth Clara, Konrat Robert, Kazimierczuk Krzysztof

Osteopontin regulates biomimetic calcium phosphate crystallization from disordered mineral layers covering apatite crystallites.

2020 Scientific reports;10(1):15722.
PMID:  32973201

Iline-Vul Taly, Nanda Raju, Mateos Borja, Hazan Shani, Matlahov Irina, Perelshtein Ilana, Keinan-Adamsky Keren, Althoff-Ospelt Gerhard, Konrat Robert, Goobes Gil

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